Pentobarbitone (Na)

Overview

Primary Characterstics

Molecular Structure of Pentobarbitone (Na)

Pentobarbitone (Na) is also known as Pentobarbital .Pentobarbitone (Na) is also known as Pentobarbital . It is of Natural origin and belongs to Barbiturate. It belongs to Chloride Channel opener (Gaba operated) pharmacological group on the basis of mechanism of action and also classified in Sedatives and Hypnotics pharmacological group.The Molecular Weight of Pentobarbitone (Na) is 248.30.

It is weakly alkaline drug, 4.07% solution of the drug is isotonic and Its pKa is 8.1.

Indications

Back to top

Pharmacokinetics

Back to top

Contraindications

Back to top

Drug Interactions

Back to top

Side Effects

Back to top

Dosage

Pentobarbitone (Na)'s dosage details are as follows:
Dose Single Dose Frequency Route Instructions

Adult Dosage

1.428 to 2.857 mg/kg2.1 (2.1425)As recommended.POAt bed time

Paedriatic Dosage (20kg)

Should not be used in children

Neonatal Dosage (3kg)

Should not be used in children

High Risk Groups

Back to top

Warning / Precautions

Pentobarbitone should not be used in patients with bronchopneumonia or status asthmaticus because it could increase respiratory depression. The drug should be used cautiously in patients with major depression or suicidal ideation, because the CNS-depressant effects of the drug can exacerbate the condition. Because of reduced renal or hepatic function, geriatric patients may require reduced doses. Pentobarbital should be used cautiously in patients with uncontrolled acute or chronic pain, with renal and the hepatic disease. It should be used with caution in patients who must perform hazardous tasks because depression of the CNS can produce effects of drowsiness and loss of mental alertness.Pentobarbitone, administered parenterally, should be used with caution in cases of hypotension, pulmonary disease, or cardiovascular disease because of possible adverse hemodynamic effects. IV administration can cause respiratory depression and should be administered slowly to avoid hypotension. It should not be prescribed in high doses for prolonged use because of the potential for psychological and physical dependence. It should not recommended for use during pregnancy because fetal abnormalities have been reported. Use of pentobarbitone in the third trimester can result in physical dependence in the neonate. If used during labor, neonates should be carefully observed for signs of respiratory depression. Premature babies are particularly sensitive to respiratory depression. Caution should be done in administering these drugs to patients with skin disease who may be predisposed to allergic reactions. Pentobarbitone is excreted into breast milk and can cause CNS depression in infants of breast-feeding mothers.Tolerance and physiological dependence can occur with pentobarbitone. Abrupt discontinuation of prolonged barbiturate therapy can result in withdrawal symptoms.

Back to top

Storage Conditions

Back to top

Interference in Pathology

Back to top

Brands / Trade Names of Pentobarbitone (Na)

Back to top

Manufacturers of Pentobarbitone (Na) in Pakistan

Back to top

Previous Drug Generic - Next Drug Generic


Suggested Pages